Compound | Class | Mechanism | In vitro IC50 | Conc. used in cells | Ref. |
---|---|---|---|---|---|
SB-415286 | Arylindole-maleimides | ATP Competitor | 78 nM | 30 μM | [44] |
AR-A014418 | Thiazole | ATP Competitor | 104 nM | 20 μM | [58] |
1-Aza kenpaullone | Benzazepinone | ATP Competitor | 18 nM | 2.5 μM | [57] |
CHIR99021 | Aminopyrimidine | ATP Competitor | 7 nM | 10 μM | [47] |
Lithium | Divalent ion | Non competitive | 2 mM | 40 mM | [41] |
TDZD-8 | Thiadiazolidinone | Non competitive | 2 μM | 10–60 μM | [70] |
Inhibitor II | Pyridyloxadiazole | - | 390 nM | 25–75 μM | [71] |
OTDZT | Thiadiazolidinone | Non competitive | 10 μM | 50–100 μM | [70] |
Inhibitor XI | Azaindolylmaleimide | ATP Competitor | 32 nM | 50 μM | [72] |